61. Synthesis of the Tetracyclic Spiro-Naphthoquinone Chartspiroton. L. Röder, K. Wurst, T. Magauer*, Org. Lett. 2024, 10.1021/acs.orglett.4c00695. (PDF-OA)


60. Synthesis of C3-epi -Virenose and Anomerically Activated Derivatives. L Röder, S. Torres Venegas, K. Wurst,  T. Magauer*, Tetrahedron Lett. 2024, accepted. (PDF-OA)


59. Synthesis of Waixenicin A: Exploring Strategies for Nine-Membered Ring Formation​. C. Steinborn, T. Huber, J. Lichtenegger, I. Plangger, D. Höfler, S. D. Schnell, L. Weisheit, P. Mayer, K. Wurst, T. Magauer*, Chem. Eur. J, 2023, 10.1002/chem.202303489. (PDF-OA).


58. Divergent Polyene Cyclization for the Total Synthesis of Greenwayodendrines, Greenwaylactams, Polysin and Polyveoline, I. Plangger, T. Pinkert, K. Wurst, T. Magauer*,  Angew. Chem., Int. Ed. 2023, 62, e202307719. (PDF-OA)


57. Total Syntheses of (+)-Waixenicin A, (+)-9-Deacetoxy-14,15-deepoxyxeniculin and (–)-Xeniafaraunol A, C. Steinborn, T. Huber, J. Lichtenegger, I. Plangger, K. Wurst, T. Magauer*,  J. Am. Chem. Soc. 2023, 145, 11811–11817. (PDF-OA)

56. Investigations into Simplified Analogues of the Herbicidal Natural Product (+)-Cornexistin, C. Steinborn, A. Tancredi, C. Habiger, C. Diederich, J. Kramer, A. Reingruber, B. Laber, J. Freigang, G. Lange, D. Schmutzler, A. Machettira, G. Besong, T. Magauer*, David M. Barber*,  Chem. Eur. J. 2023, 29, e202300199. (PDF-OA)

55. Total Synthesis of the Dihydrooxepine-Spiroisoxazoline Natural Product Psammaplysin A, J. Paciorek, D. Hoefler, K. R. Sokol, K. Wurst, T. Magauer*,  J. Am. Chem. Soc. 2022, 144, 19704–19708. (PDF-OA)
ChemRxiv DOI: 10.26434/chemrxiv-2022-px26h.


54. Short, Divergent and Enantioselective Total Synthesis of Bioactive ent-Pimaranes. I. Plangger, K. Wurst, T. Magauer*, Org. Lett. 2022, 24, 7151−7156. (PDF-OA)


53. KS0365, a novel activator of the transient receptor potential vanilloid 3 (TRPV3) channel, accelerates keratinocyte migration. M. Maier, S. Olthoff, K. Hill, C. Zosel, T. Magauer, L. A. Wein, M. Schaefer, Br J Pharmacol. 2022179, 5290–5304. (PDF-OA)


52. A General Entry to Ganoderma Meroterpenoids: Synthesis of Lingzhiol via Photoredox Catalysis. A. Rode, K. Wurst, T. Magauer*, ChemRxiv 2022, DOI: 10.26434/chemrxiv-2022-svqft. (PDF-OA)


51. Total Synthesis and Late-Stage C–H Oxidations of ent-Trachylobane Natural Products. L. A. Wein, K. Wurst, T. Magauer*, Angew. Chem., Int. Ed. 202261, e202113829 (VIP). (PDF-OA)


50. Ring-Expansion of 1-Indanones to 2-Halo-1-naphthols as an Entry Point to Gilvocarcin Natural Products. I. Zamarija, B. Marsh, T. Magauer*, Org. Lett. 202123, 9221−9226(PDF-OA)


49. Bifunctional Polyene Cyclizations: Synthetic Studies on Pimarane Natural Products. J. M. Feilner, I. Plangger, T. Magauer*, Chem. Eur. J. 2021, 27, 12410–12421. (PDF-OA)


48. Total Synthesis of Oxepin and Dihydrooxepin Containing Natural Products. K. R. Sokol, T. Magauer*, Synthesis 202153, 4187-4202. (PDF)


47. Synthesis of Pyrroles via Consecutive 6π-Electrocyclization/Ring-Contraction of Sulfilimines. F.-L. Haut, N. Feichtinger; I. Plangger, L. Wein, M. Müller, T.-N. Streit, K. Wurst,  M. Podewitz, T. Magauer*, J. Am. Chem. Soc. 2021143, 9002–9008. (PDF-OA)


46. Evolution of a Strategy for the Total Synthesis of (+)-Cornexistin. R. E. Wildermuth, C. Steinborn, D. M. Barber, K. S. Mühlfenzl, M. Kendlbacher, P. Mayer, K. Wurst, T. Magauer*, Chem. Eur. J. 2021, 27, 1218112189. (PDF-OA)


45. The 2nd Alpine Winter Conference on Medicinal and Synthetic Chemistry. A. Ciulli, L. Hamann, W. Jahnke, A. Kalgutkar, T. Magauer, T. Ritter, V. Steadman, S. D. Williams, G. Winter, K. Hoegenauer, K. H. Krawinkler, A. F. Stepan, ChemMedChem 2021, 16, 2417–24232. (PDF-OA)

44. Beyond the Isoprene Pattern: Bifunctional Polyene Cyclizations. J. M. Feilner, F.-L. Haut, T. Magauer*, Chem. Eur. J. 202127, 7017–7021. (PDF-OA) (Concept Article)


43. Rapid Assembly of Tetrasubstituted Furans via Pummerer-type Rearrangement. F.-L. Haut, C. Habiger, L. A. Wein, K. Wurst, M. Podewitz*, T. Magauer* J. Am. Chem. Soc. 2021, 143, 1216–1223. (PDF-OA)


42. Synthesis of Vicinal Quaternary All-Carbon Centers via Acid-catalyzed Cycloisomerization of Neopentylic Epoxides.
M. Schmid, K. R. Sokol, L. A. Wein, S. Torres Venegas, C. Meisenbichler, K. Wurst, M. Podewitz,  T. Magauer*, Org. Lett. 2020, 22, 6526–6531. (PDF-OA).


41. Total Synthesis of (+)-Cornexistin.
C. Steinborn, R. E. Wildermuth, D. M. Barber,  T. Magauer*, Angew. Chem., Int. Ed. 2020, 59, 17282–17285. (PDF-OA)


40. A Transannular Polyene Tetracyclization for the Rapid Construction of the Pimarane Framework.
J. M. Feilner, K. Wurst,  T. Magauer*, Angew. Chem., Int. Ed. 2020, 59, 12436–12439. (PDF-OA)


39. Synthesis of (–)-Mitrephorone A via a Bio-inspired Late Stage C–H Oxidation of (–)-Mitrephorone B.
L. A. Wein, K. Wurst, P. Angyal, L. Weisheit, T. Magauer*, J. Am. Chem. Soc. 2019, 141, 19589–19593. (PDF-OA)

2020_Mitrephorone B and A

38. A Synthetic Entry to Polyfunctionalized Molecules through the [3+2]-Cycloaddition of Thiocarbonyl Ylides.
F.-L. Haut, C. Habiger, K. Speck, K. Wurst, P. Mayer, J. N. Korber, T. Müller, T. Magauer*, J. Am. Chem. Soc. 2019, 141, 13352−13357. (PDF-OA)


37. Ring-Expansion Approaches for the Total Synthesis of Salimabromide.
M. Schmid, A. Grossmann, P. Mayer, T. Müller, T. Magauer*, Tetrahedron 2019, 75, 3195–3215. (PDF-OA)


36. Total Synthesis of Salimabromide, a Tetracyclic Polyketide from a Marine Myxobacterium.
M. Schmid, A. Grossmann, K. Wurst, T. Magauer*, J. Am. Chem. Soc. 2018, 140, 8444–8447. (PDF-OA)

This work was highlighted as Synfact of the Month: E. M. Carreira, N. Sievertsen, Synfacts 2018, 14, 0887. (PDF)


35. A Negishi cross-coupling reaction enables the total synthesis of (+)-stachyflin.
F.-L. Haut, K. Speck, R. Wildermuth, K. Möller, P. Mayer, T. Magauer*, Tetrahedron 2018, 74, 3348–3357. (PDF)


34. 9-Membered Carbocycles: Strategies and Tactics for their Synthesis.
T. Huber, R. Wildermuth, T. Magauer*, Chem. Eur. J. 2018, 24, 12107–12120. (PDF-OA)


33. De Novo Synthesis of Benzannelated Heterocycles.
J. Feierfeil, T. Magauer*, Chem. Eur. J. 2018, 24, 1455–1458. (PDF)


32. A Modular Synthesis of Tetracyclic Meroterpenoid Antibiotics.
R. Wildermuth, K. Speck, F.-L. Haut, P. Mayer, B. Karge, M. Brönstrup, T. Magauer*, Nat. Commun. 2017, 8, 2083. (PDF-OA)


31. Development of a β-C–H Bromination Approach Towards the Synthesis of Jerantinine E.
T. Huber, T. Unzner, C. Gerlinger, T. Magauer*J. Org. Chem. 2017, 82, 7410–7419. (PDF)


30. Dyotropic Rearrangements in Natural Product Synthesis and Biosynthesis.
C. L. Hugelshofer, T. Magauer*Nat. Prod. Rep2017, 34, 228–234. (Highlight) (PDF)

29. Bioinspired Total Syntheses of Terpenoids.
C. L. Hugelshofer, T. Magauer*, Org. Biomol. Chem. 201715, 12–16. (Perspective) (PDF)

28. Evolution of a Polyene Cyclization Cascade for the Total Synthesis of (–)-Cyclosmenospongine.
K. Speck, T. Magauer*, Chem. Eur. J. 2017, 23, 1157–1165. (HOT PAPER) (PDF)

27. Convergent Assembly of the Tetracyclic Meroterpenoid (–)-Cyclosmenospongine via a Non-Biomimetic Polyene Cyclization.
K. Speck, R. Wildermuth, T. Magauer*, Angew. Chem. Int. Ed. 2016, 55, 14131–14135. (PDF)

This work was highlighted in SYNFACTS: E. M. Carreira, P. Sondermann, Synfacts 2017, 13, 5.

26. A Divergent Approach to the Marine Diterpenoids (+)-Dictyoxetane and (+)-Dolabellane V.
C. L. Hugelshofer, T. Magauer*Chem. Eur. J. 201622, 15125–15136. (PDF)

25. Rapid Access to Orthogonally Functionalized Naphthalenes: Application to the Total Synthesis of the Anticancer Agent Chartarin.
T. A. Unzner, A. Grossmann, T. Magauer*Angew. Chem., Int. Ed. 2016, 55, 9763–9767. (HOT PAPER) (PDF)

24. A Bioinspired Cyclization Sequence Enables the Asymmetric Total Synthesis of Dictyoxetane.
C. L. Hugelshofer, T. Magauer*J. Am. Chem. Soc. 2016, 138, 6420–6423. (PDF)

This work was highlighted in SYNFACTS: E. M. Carreira, H. Wolleb, Synfacts 201612, 771. 

23. Gold(I)-Catalyzed Enyne Cyclizations: Studies Towards the Total Synthesis of (+)-Aureol.
R. Wildermuth, K. Speck, T. Magauer*, Synthesis, 2016, 48, 1814–1824. (PDF)

22. Trihaloethenes as Versatile Building Blocks for Organic Synthesis.
A. Grossmann, T. Magauer*, Org. Biomol. Chem. 2016, 14, 5377–5389 (Review). (PDF)


21. Synthesis of Xenia diterpenoids and related metabolites isolated from marine organisms.
T. Huber, L. Weisheit, T. Magauer*, Beilstein J. Org. Chem. 201511, 2521–2539 (Review). (PDF)

20. Ring Opening of Bicyclic[3.1.0]hexan-2-ones: A Versatile Synthetic Platform for the Construction of Substituted Benzoates.
J. Feierfeil, A. Grossmann, T. Magauer*, Angew. Chem., Int. Ed. 2015, 54, 11835–11838. (PDF)

19. The 50th EUCHEM Conference on Stereochemistry (Bürgenstock Conference 2015).
A. Adibekian, T. Magauer*, Chimia, 201569, 485–487 (Conference Report). (PDF)

18. Sequential O–H/C–H Bond Insertion of Phenols initiated by the Gold(I)-Catalyzed Cyclization of 1-Bromo-1,5-Enynes.
K. Speck, K. Karaghiosoff, T. Magauer*, Org. Lett. 2015, 17, 1982–1985. (PDF)

17. Total Synthesis of the Leucosceptroid Family of Natural Products.
C. L. Hugelshofer, T. Magauer*, J. Am. Chem. Soc. 2015, 137, 3807–3810. (PDF)

16. Experimental Studies on the Selective beta-C-H Halogenation of Enones.
T. Huber, J. Rickmeier, D. Kaiser, T. Magauer*, J. Org. Chem. 2015, 80, 2281–2294. (PDF)

15. Chemical Synthesis of Antifeedant Leucosceptroids.
C. L. Hugelshofer, K. Speck, A. S. Grossmann, T. Magauer*, Beilstein TV, 2015. Beilstein Video

14. Carbon-Fluorine Bond Activation for the Synthesis of Functionalized Molecules.
T. A. Unzner, T. Magauer*Tetrahedron Lett. 2015, 56, 877–883 (Review). (PDF)

13. Strategies for the Synthesis of Antifeedant Leucosceptroid Natural Products.
C. L. Hugelshofer, T. Magauer*Synlett 2015, 26, 572–579 (Review)(PDF)

12. Unraveling the Metabolic Pathway in Leucosceptrum canum by Isolation of New Defensive Leucosceptroid Degradation Products and Biomimetic Model Synthesis.
S.-H. Luo, C. L. Hugelshofer, J. Hua, S.-X. Jing, C.-H. Li, Y. Liu, X.-N. Li, X. Zhao, T. Magauer*, S.-H. Li*, Org. Lett. 2014, 16, 6416–6419.  (PDF)


11. A General Entry to Antifeedant Sesterterpenoids: Total Synthesis of (+)-Norleucosceptroid A, (–)-Norleucosceptroid B, and (–)-Leucosceptroid K.
C. L. Hugelshofer, T. Magauer*Angew. Chem., Int. Ed. 2014, 53, 11351–11355.  (PDF)

This work was selected as SYNFACT of the month: E. M. Carreira, M. Westphal, Synfacts 201410, 1233.

10. Crystalline guanine adducts of natural and synthetic trioxacarcins suggest a common biological mechanism and reveal a basis for the instability of trioxacarcin.
K. Pröpper, B. Dittrich, D. J. Smaltz, T. Magauer, A. G. Myers, Biorg. Med. Chem. Lett. 2014, 24, 4410–4413.  (PDF)

9. A transition metal-free synthesis of fluorinated naphthols.
J. Hammann, T. Unzner, T. Magauer*, Chem. Eur. J. 2014, 20, 6733–6738.  (PDF)

This work was highlighted in SYNFACTS: P. Knochel, D. Haas, Synfacts 2014, 10, 853.

8. High-Pressure Transformations in Natural Product Synthesis.
C. L. Hugelshofer, T. Magauer*Synthesis 2014, 46, 1279–1296 (Review). (PDF)


7. The Chemistry of Isoindole Natural Products.
K. Speck, T. Magauer*Beilstein J. Org. Chem. 20139, 2048–2078 (Review). (PDF)

6. Component-Based Syntheses of Trioxacarcin A, DC-45-A1, and Structural Analogs.
T. Magauer, D. Smaltz, A. G. Myers, Nat. Chem. 20135, 886–893. (PDF)


5. Short and Efficient Synthetic Route to Methyl α-Trioxacarcinoside B and Anomerically Activated Derivatives.
T. Magauer, A. G. Myers, Org. Lett. 201113, 5584–5587. (PDF)


4. In Pursuit of a Competitive Target: the Total Synthesis of the Antibiotic Kendomycin.
H. J. Martin, T. Magauer, J. Mulzer, Angew. Chem., Int. Ed. 2010, 49, 5614–5626 (Review). (PDF)


3. Ring Closing Metathesis and Photo–Fries Reaction for the Construction of the Ansamycin Antibiotic Kendomycin. Development of a Protecting Group Free Oxidative Endgame.
T. Magauer, H. J. Martin, J. Mulzer, Chem. Eur. J. 2010, 16, 507–519. (PDF)


2. Total Synthesis of (+)–Echinopine A and B: Determination of Absolute Stereochemistry.
T. Magauer*, J. Mulzer, K. Tiefenbacher,* Org. Lett. 200911, 5306–5309. (PDF)


1. Total Synthesis of the Antibiotic Kendomycin by Macrocyclization via Photo–Fries Rearrangement and Ring Closing Metathesis.
T. Magauer, H. J. Martin, J. Mulzer, Angew. Chem., Int. Ed. 200948, 6032–6036. (PDF)




Trioxacarcins and Uses Thereof,  Andrew G. Myers, Nicholas E. Hill, Jakub Svenda, Robert T. Yu, Daniel J. Smaltz, and Thomas Magauer, International PCT Patent Application No. PCT/US2011/029343, filed March 22, 2011.

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