Books

Publications

 

49. Bifunctional Polyene Cyclizations: Synthetic Studies on Pimarane Natural Products. J. M. Feilner, I. Plangger, T. Magauer*, Chem. Eur. J. 2021, 10.1002/chem.202101926. (PDF-OA)

2021_cej_pimarendiolfull

48. Total Synthesis of Oxepin and Dihydrooxepin Containing Natural Products. K. R. Sokol, T. Magauer*, Synthesis 202110.1055/s-0037-1610776. (PDF)

2021_synthesisoxepin

47. Synthesis of Pyrroles via Consecutive 6π-Electrocyclization/Ring-Contraction of Sulfilimines. F.-L. Haut, N. Feichtinger; I. Plangger, L. Wein, M. Müller, T.-N. Streit, K. Wurst,  M. Podewitz, T. Magauer*, J. Am. Chem. Soc. 2021143, 9002–9008. (PDF-OA)

2021_Pyrroles_JACS

46. Evolution of a Strategy for the Total Synthesis of (+)-Cornexistin. R. E. Wildermuth, C. Steinborn, D. M. Barber, K. S. Mühlfenzl, M. Kendlbacher, P. Mayer, K. Wurst, T. Magauer*, Chem. Eur. J. 202110.1002/chem.202101849. (PDF-OA)

2021_CEJ_Cornexistin

45. The 2nd Alpine Winter Conference on Medicinal and Synthetic Chemistry. A. Ciulli, L. Hamann, W. Jahnke, A. Kalgutkar, T. Magauer, T. Ritter, V. Steadman, S. D. Williams, G. Winter, K. Hoegenauer, K. H. Krawinkler, A. F. Stepan, ChemMedChem 2021, 1610.1002/cmdc.202100372. (PDF-OA)

44. Beyond the Isoprene Pattern: Bifunctional Polyene Cyclizations. J. M. Feilner, F.-L. Haut, T. Magauer*, Chem. Eur. J. 202127, 7017–7021. (PDF-OA) (Concept Article)

2021_conceptPolyene


43. Rapid Assembly of Tetrasubstituted Furans via Pummerer-type Rearrangement. F.-L. Haut, C. Habiger, L. A. Wein, K. Wurst, M. Podewitz*, T. Magauer* J. Am. Chem. Soc. 2021, 143, 1216–1223. (PDF-OA)

2021_Furans_JACS


42. Synthesis of Vicinal Quaternary All-Carbon Centers via Acid-catalyzed Cycloisomerization of Neopentylic Epoxides.
M. Schmid, K. R. Sokol, L. A. Wein, S. Torres Venegas, C. Meisenbichler, K. Wurst, M. Podewitz,  T. Magauer*, Org. Lett. 2020, 22, 6526–6531. (PDF-OA).

2020_Org_lett_Tetralins



41. Total Synthesis of (+)-Cornexistin.
C. Steinborn, R. E. Wildermuth, D. M. Barber,  T. Magauer*, Angew. Chem., Int. Ed. 2020, 59, 17282–17285. (PDF-OA)

2020_cornexisitin_toc_


40. A Transannular Polyene Tetracyclization for the Rapid Construction of the Pimarane Framework.
J. M. Feilner, K. Wurst,  T. Magauer*, Angew. Chem., Int. Ed. 2020, 59, 12436–12439. (PDF-OA)

 2020_pimarane_toc_revised


39. Synthesis of (–)-Mitrephorone A via a Bio-inspired Late Stage C–H Oxidation of (–)-Mitrephorone B.
L. A. Wein, K. Wurst, P. Angyal, L. Weisheit, T. Magauer*, J. Am. Chem. Soc. 2019, 141, 19589–19593. (PDF-OA)

2020_Mitrephorone B and A


38. A Synthetic Entry to Polyfunctionalized Molecules through the [3+2]-Cycloaddition of Thiocarbonyl Ylides.
F.-L. Haut, C. Habiger, K. Speck, K. Wurst, P. Mayer, J. N. Korber, T. Müller, T. Magauer*, J. Am. Chem. Soc. 2019, 141, 13352−13357. (PDF-OA)

2019_JACS_High_pressure


37. Ring-Expansion Approaches for the Total Synthesis of Salimabromide.
M. Schmid, A. Grossmann, P. Mayer, T. Müller, T. Magauer*, Tetrahedron 2019, 75, 3195–3215. (PDF-OA)

2019_Tet_Salimabromide


36. Total Synthesis of Salimabromide, a Tetracyclic Polyketide from a Marine Myxobacterium.
M. Schmid, A. Grossmann, K. Wurst, T. Magauer*, J. Am. Chem. Soc. 2018, 140, 8444–8447. (PDF-OA)

This work was highlighted as Synfact of the Month: E. M. Carreira, N. Sievertsen, Synfacts 2018, 14, 0887. (PDF)

2018_JACS_salimabromide


35. A Negishi cross-coupling reaction enables the total synthesis of (+)-stachyflin.
F.-L. Haut, K. Speck, R. Wildermuth, K. Möller, P. Mayer, T. Magauer*, Tetrahedron 2018, 74, 3348–3357. (PDF)

 2018_tetrahedron_stachyflin_new


34. 9-Membered Carbocycles: Strategies and Tactics for their Synthesis.
T. Huber, R. Wildermuth, T. Magauer*, Chem. Eur. J. 2018, 24, 12107–12120. (PDF-OA)

 9-membered-rings


33. De Novo Synthesis of Benzannelated Heterocycles.
J. Feierfeil, T. Magauer*, Chem. Eur. J. 2018, 24, 1455–1458. (PDF)

Heterocycles_Johannes


32. A Modular Synthesis of Tetracyclic Meroterpenoid Antibiotics.
R. Wildermuth, K. Speck, F.-L. Haut, P. Mayer, B. Karge, M. Brönstrup, T. Magauer*, Nat. Commun. 2017, 8, 2083. (PDF-OA)

 2017_Nat_Commun_Meroterpenoids


31. Development of a β-C–H Bromination Approach Towards the Synthesis of Jerantinine E.
T. Huber, T. Unzner, C. Gerlinger, T. Magauer*J. Org. Chem. 2017, 82, 7410–7419. (PDF)

JOC_Tatjana_Tesi_Christa


30. Dyotropic Rearrangements in Natural Product Synthesis and Biosynthesis.
C. L. Hugelshofer, T. Magauer*Nat. Prod. Rep2017, 34, 228–234. (Highlight) (PDF)



29. Bioinspired Total Syntheses of Terpenoids.
C. L. Hugelshofer, T. Magauer*, Org. Biomol. Chem. 201715, 12–16. (Perspective) (PDF)



28. Evolution of a Polyene Cyclization Cascade for the Total Synthesis of (–)-Cyclosmenospongine.
K. Speck, T. Magauer*, Chem. Eur. J. 2017, 23, 1157–1165. (HOT PAPER) (PDF)



27. Convergent Assembly of the Tetracyclic Meroterpenoid (–)-Cyclosmenospongine via a Non-Biomimetic Polyene Cyclization.
K. Speck, R. Wildermuth, T. Magauer*, Angew. Chem. Int. Ed. 2016, 55, 14131–14135. (PDF)


This work was highlighted in SYNFACTS: E. M. Carreira, P. Sondermann, Synfacts 2017, 13, 5.


26. A Divergent Approach to the Marine Diterpenoids (+)-Dictyoxetane and (+)-Dolabellane V.
C. L. Hugelshofer, T. Magauer*Chem. Eur. J. 201622, 15125–15136. (PDF)



25. Rapid Access to Orthogonally Functionalized Naphthalenes: Application to the Total Synthesis of the Anticancer Agent Chartarin.
T. A. Unzner, A. Grossmann, T. Magauer*Angew. Chem., Int. Ed. 2016, 55, 9763–9767. (HOT PAPER) (PDF)



24. A Bioinspired Cyclization Sequence Enables the Asymmetric Total Synthesis of Dictyoxetane.
C. L. Hugelshofer, T. Magauer*J. Am. Chem. Soc. 2016, 138, 6420–6423. (PDF)

This work was highlighted in SYNFACTS: E. M. Carreira, H. Wolleb, Synfacts 201612, 771. 


23. Gold(I)-Catalyzed Enyne Cyclizations: Studies Towards the Total Synthesis of (+)-Aureol.
R. Wildermuth, K. Speck, T. Magauer*, Synthesis, 2016, 48, 1814–1824. (PDF)



22. Trihaloethenes as Versatile Building Blocks for Organic Synthesis.
A. Grossmann, T. Magauer*, Org. Biomol. Chem. 2016, 14, 5377–5389 (Review). (PDF)

 


21. Synthesis of Xenia diterpenoids and related metabolites isolated from marine organisms.
T. Huber, L. Weisheit, T. Magauer*, Beilstein J. Org. Chem. 201511, 2521–2539 (Review). (PDF)


20. Ring Opening of Bicyclic[3.1.0]hexan-2-ones: A Versatile Synthetic Platform for the Construction of Substituted Benzoates.
J. Feierfeil, A. Grossmann, T. Magauer*, Angew. Chem., Int. Ed. 2015, 54, 11835–11838. (PDF)



19. The 50th EUCHEM Conference on Stereochemistry (Bürgenstock Conference 2015).
A. Adibekian, T. Magauer*, Chimia, 201569, 485–487 (Conference Report). (PDF)


18. Sequential O–H/C–H Bond Insertion of Phenols initiated by the Gold(I)-Catalyzed Cyclization of 1-Bromo-1,5-Enynes.
K. Speck, K. Karaghiosoff, T. Magauer*, Org. Lett. 2015, 17, 1982–1985. (PDF)



17. Total Synthesis of the Leucosceptroid Family of Natural Products.
C. L. Hugelshofer, T. Magauer*, J. Am. Chem. Soc. 2015, 137, 3807–3810. (PDF)



16. Experimental Studies on the Selective beta-C-H Halogenation of Enones.
T. Huber, J. Rickmeier, D. Kaiser, T. Magauer*, J. Org. Chem. 2015, 80, 2281–2294. (PDF)



15. Chemical Synthesis of Antifeedant Leucosceptroids.
C. L. Hugelshofer, K. Speck, A. S. Grossmann, T. Magauer*, Beilstein TV, 2015. Beilstein Video


14. Carbon-Fluorine Bond Activation for the Synthesis of Functionalized Molecules.
T. A. Unzner, T. Magauer*Tetrahedron Lett. 2015, 56, 877–883 (Review). (PDF)


13. Strategies for the Synthesis of Antifeedant Leucosceptroid Natural Products.
C. L. Hugelshofer, T. Magauer*Synlett 2015, 26, 572–579 (Review)(PDF)



12. Unraveling the Metabolic Pathway in Leucosceptrum canum by Isolation of New Defensive Leucosceptroid Degradation Products and Biomimetic Model Synthesis.
S.-H. Luo, C. L. Hugelshofer, J. Hua, S.-X. Jing, C.-H. Li, Y. Liu, X.-N. Li, X. Zhao, T. Magauer*, S.-H. Li*, Org. Lett. 2014, 16, 6416–6419.  (PDF)

 


11. A General Entry to Antifeedant Sesterterpenoids: Total Synthesis of (+)-Norleucosceptroid A, (–)-Norleucosceptroid B, and (–)-Leucosceptroid K.
C. L. Hugelshofer, T. Magauer*Angew. Chem., Int. Ed. 2014, 53, 11351–11355.  (PDF)

This work was selected as SYNFACT of the month: E. M. Carreira, M. Westphal, Synfacts 201410, 1233.


10. Crystalline guanine adducts of natural and synthetic trioxacarcins suggest a common biological mechanism and reveal a basis for the instability of trioxacarcin.
K. Pröpper, B. Dittrich, D. J. Smaltz, T. Magauer, A. G. Myers, Biorg. Med. Chem. Lett. 2014, 24, 4410–4413.  (PDF)


9. A transition metal-free synthesis of fluorinated naphthols.
J. Hammann, T. Unzner, T. Magauer*, Chem. Eur. J. 2014, 20, 6733–6738.  (PDF)

This work was highlighted in SYNFACTS: P. Knochel, D. Haas, Synfacts 2014, 10, 853.



8. High-Pressure Transformations in Natural Product Synthesis.
C. L. Hugelshofer, T. Magauer*Synthesis 2014, 46, 1279–1296 (Review). (PDF)

 


7. The Chemistry of Isoindole Natural Products.
K. Speck, T. Magauer*Beilstein J. Org. Chem. 20139, 2048–2078 (Review). (PDF)



6. Component-Based Syntheses of Trioxacarcin A, DC-45-A1, and Structural Analogs.
T. Magauer, D. Smaltz, A. G. Myers, Nat. Chem. 20135, 886–893. (PDF)

 

5. Short and Efficient Synthetic Route to Methyl α-Trioxacarcinoside B and Anomerically Activated Derivatives.
T. Magauer, A. G. Myers, Org. Lett.201113, 5584–5587. (PDF)

 

4. In Pursuit of a Competitive Target: the Total Synthesis of the Antibiotic Kendomycin.
H. J. Martin, T. Magauer, J. Mulzer, Angew. Chem., Int. Ed. 2010, 49, 5614–5626 (Review). (PDF)

 

3. Ring Closing Metathesis and Photo–Fries Reaction for the Construction of the Ansamycin Antibiotic Kendomycin. Development of a Protecting Group Free Oxidative Endgame.
T. Magauer, H. J. Martin, J. Mulzer, Chem. Eur. J. 2010, 16, 507–519. (PDF)

 

2. Total Synthesis of (+)–Echinopine A and B: Determination of Absolute Stereochemistry.
T. Magauer*, J. Mulzer, K. Tiefenbacher,* Org. Lett.200911, 5306–5309. (PDF)

 

1. Total Synthesis of the Antibiotic Kendomycin by Macrocyclization via Photo–Fries Rearrangement and Ring Closing Metathesis.
T. Magauer, H. J. Martin, J. Mulzer, Angew. Chem., Int. Ed. 200948, 6032–6036. (PDF)

 

 

Patents

Trioxacarcins and Uses Thereof,  Andrew G. Myers, Nicholas E. Hill, Jakub Svenda, Robert T. Yu, Daniel J. Smaltz, and Thomas Magauer, International PCT Patent Application No. PCT/US2011/029343, filed March 22, 2011.

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